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Description

A reversible and ATP-competitive inhibitor of protein kinase C (Ki = 10 nM). Inhibits protein kinase A at much higher concentrations (Ki = 2 µ,M). An enhanced water soluble form of Bisindolylmaleimide I (Cat. No. 203290)., An enhanced water-soluble form of Bisindolylmaleimide I (Cat. No. 203290). A reversible and ATP-competitive inhibitor of protein kinase C (Ki = 10 nM). May inhibit protein kinase A at much higher concentrations (Ki = 2 µ,M).

Structure formula

GF 109203X hydrochloride

Contents

Miscellaneous

Certificate of Analysis (specimen)

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Product data sheet

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