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Beschreibung

A reversible and ATP-competitive inhibitor of protein kinase C (Ki = 10 nM). Inhibits protein kinase A at much higher concentrations (Ki = 2 µ,M). An enhanced water soluble form of Bisindolylmaleimide I (Cat. No. 203290)., An enhanced water-soluble form of Bisindolylmaleimide I (Cat. No. 203290). A reversible and ATP-competitive inhibitor of protein kinase C (Ki = 10 nM). May inhibit protein kinase A at much higher concentrations (Ki = 2 µ,M).

Strukturformel

GF 109203X hydrochloride

Inhalte

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