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Description

A highly potent and selective non-alkaloid positive allosteric modulator of Kappa-opioid receptors (Ki = 4.3 nM and 16 nM for native and cloned kappa-opioid receptors, respectively). Also acts as a D2DR partial agonist (Ki = 5-10 nM). Used in studies of addition.

Structure formula

Salvinorin A

Contents

Miscellaneous

Certificate of Analysis (specimen)

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Product data sheet

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