Item no.
SAF-123850-25MG
CAS Number
[4906-68-7]
Unit
1 x 25 mg
Molecular formula
C13H9BrO3
Molecular weight
293,11
Shipment details
No Dangerous Good
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Description
A cell-permeable salicylic acid compound that acts as a highly potent, active-site directed and substrate competitive AKR1C1 inhibitor (Ki = 4 nM) with moderate to excellent selectivity over AKR1C2, AKR1C3 and AKR1C4 (Ki = 0.087, 4.2 and 18.2 µ,M, respectively). Shown to inhibit the metabolism of progesterone by AKR1C1 (IC50 = 460 nM in AKR1C1 overexpressing BAECs).
Structure formula
Contents
Miscellaneous
Certificate of Analysis (specimen)
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Product data sheet
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