Artikelnr.
SAF-5057230001
CAS-Nummer
[125941-87-9]
Einheit
EA
Molekularformel
C17H19Cl2NO
Molekulargewicht
324,24
Transportdaten
No Dangerous Good /not restricted
A highly potent and selective dopamine D1-like receptor antagonist with a Ki of 0.2 and 0.3 nM for the D1 and D5 dopamine receptor subtypes, respectively. Also an agonist at 5-HT1C and 5-HT2C receptors in vitro (Ki values are 6.3 nM and 9.3 nM respectively).
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